In the competitive world of athletics and bodybuilding, the quest for enhanced performance and physique often extends beyond traditional training and nutrition. Athletes and fitness enthusiasts alike are increasingly turning to a variety of non-steroidal, orally administered performance-enhancing drugs (PEDs) that promise benefits like increased strength, endurance, and cognitive function. These substances range from compounds that mimic the effects of anabolic steroids to others that stimulate fat loss, enhance alertness, or even mask the use of other banned substances. This section explores a selection of such PEDs, each with its unique properties and applications.

Expanded Overview of Non-Steroidal Oral PEDs

Selective Androgen Receptor Modulators (SARMs):

Examples: Ostarine (MK-2866), Andarine (S4), Ligandrol (LGD-4033).

Benefits: Mimic the muscle growth effects of anabolic steroids.

Usage: Primarily in muscle building and fat loss, targeting specific androgen receptors in muscle and bone tissues.

Side Effects: Often marketed as having fewer side effects than traditional steroids, but long-term effects are still under research.

Stimulants

Examples: Amphetamines, Methylhexanamine (in pre-workout supplements), Modafinil.

Benefits: Enhance alertness, reduce fatigue, and improve concentration.

Usage: Common in sports requiring high levels of endurance and focus.

Side Effects: Can include heart palpitations, insomnia, and increased risk of cardiovascular events.

Beta-2 Agonists:

Examples: Clenbuterol, Albuterol.

Benefits: Promote fat loss and muscle gain.

Usage: Initially for asthma, but now used for its fat-burning and anabolic properties.

Side Effects: Can lead to cardiac issues, tremors, and anxiety.