Aromatase Inhibitor
Active Ingredient:Exemestane
Tablet Count: 50 Tablets
Half-Life: 24 Hours
Classification: Aromatase Inhıbıtor
Dosage: 12.5-25 mg per day
Acne: Low
Water Retention: Low
Hepatotoxicity: Low
Aromatization: Prevents
Exemestane, marketed under the brand name Aromasin, is a potent aromatase inhibitor widely used in bodybuilding and athletic circles to manage estrogen levels and enhance muscle definition. Bodybuilders and athletes rely on Exemestane during and after anabolic steroid cycles to prevent estrogenic side effects and maintain optimal hormone balance.
Mechanism of Action:
Exemestane works by irreversibly binding to the aromatase enzyme, which is responsible for converting androgens (like testosterone) into estrogen in the body. By inhibiting this enzyme, Exemestane effectively reduces estrogen levels. This reduction is crucial for managing estrogenic side effects such as gynecomastia (development of breast tissue in men), water retention, and fat gain. The drug’s action helps in preserving muscle definition and achieving a leaner physique.
Usage and Dosage
The standard dosage of Exemestane is 12.5-25 mg daily, depending on the user’s individual needs and the extent of estrogen-related side effects. For those on an anabolic steroid cycle or undergoing post-cycle therapy (PCT), Exemestane is typically taken daily to maintain effective estrogen control. It’s important to note that excessive use of aromatase inhibitors can lead to overly suppressed estrogen levels, potentially affecting joint health and other physiological functions.